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Drug reference

abiraterone acetate

CYP17A1 inhibitor · Steroidogenesis inhibitor

CYP17A1 inhibitorSteroidogenesis inhibitor
CDSCO approved
EXCRETION
not curated
INTERACTIONS
none in our sources
PREGNANCY
not curated

Mechanism

Abiraterone acetate is a CYP17A1 inhibitor.

Indications

prostate cancerendogenous cushing syndrome (under evaluation)reduction of adrenal androgen production in congenital adrenal hyperplasia (under evaluation)

Related guidelines

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Sources: Goodman & Gilman 14e·Verified: 2026-05-10 · House clinical team