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Drug reference

cyproheptadine

Piperidine (H1 Antagonist) · Antiallergic, Antiserotonin, Antipruritic

Piperidine (H1 Antagonist)Antiallergic, Antiserotonin, Antipruritic
CDSCO approved
EXCRETION
—
not curated
INTERACTIONS
6 major
SEVERE in our sources
PREGNANCY
—
not curated
Top interactionssee all 6 →
  • DextropropoxypheneSevereDatabaseDDInter
  • Potassium ChlorideSevereDatabaseDDInter
  • Potassium CitrateSevereDatabaseDDInter
  • Sodium OxybateSevereDatabaseDDInter

Mechanism

Not yet extracted

Indications

appetite stimulation (off label in anorectic/convalescent patients)idiopathic pruritus

Dosing

Adult
4 mg oral

Side effects

Common
sedationdiminished alertnesslight headednessmotor incoordinationfatiguetendency to fall asleepappetite stimulating effectdry mouthalteration of bowel movementurinary hesitancyblurring of vision

Drug interactions

Dextropropoxyphene
Severe
Database

Clinical effect not specified

Source: DDInter

Potassium Chloride
Severe
Database

.

Source: DDInter

Potassium Citrate
Severe
Database

Clinical effect not specified

Source: DDInter

Sodium Oxybate
Severe
Database

Clinical effect not specified

Source: DDInter

Topiramate
Severe
Database

Clinical effect not specified

Source: DDInter

Zonisamide
Severe
Database

Clinical effect not specified

Source: DDInter

6 additional unreviewed or low-confidence interactions hidden because their provenance or source detail is insufficient.

Other Piperidine (H1 Antagonist) drugs

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Textbook-sourced·Sources: KD Tripathi 7e, Goodman & Gilman 14e·Updated: 2026-05-10