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Drug reference

relatlimab

human IgG4, LAG3 inhibitor, immune checkpoint inhibitor · anticancer, immunomodulator

human IgG4, LAG3 inhibitor, immune checkpoint inhibitoranticancer, immunomodulator
CDSCO approved
EXCRETION
not curated
INTERACTIONS
none in our sources
PREGNANCY
not curated

Mechanism

Relatlimab is a human IgG4 that targets LAG3 (lymphocyte activation gene 3).

Indications

untreated advanced melanoma (in combination with nivolumab)first-line treatment of advanced melanoma (in combination with nivolumab)activity after progression on other checkpoint inhibitorsinvestigated in the neoadjuvant setting for palpable nodal disease

Side effects

Common
skin rashdiarrhea (sometimes severe, life-threatening colitis)
Serious
  • thyroiditis
  • hypophysitis
  • hepatitis
  • nephritis
  • pneumonitis
  • myocarditis
  • neuritis

Related guidelines

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Sources: Goodman & Gilman 14e, Harrison 22e·Verified: 2026-05-10 · House clinical team