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tocopherol

Fat-soluble vitamin · Vitamin supplement

Fat-soluble vitaminVitamin supplement
CDSCO approved
EXCRETION
not curated
INTERACTIONS
none in our sources
PREGNANCY
not curated

Mechanism

Vitamin E (α-tocopherol) acts as an antioxidant, protecting unsaturated lipids in cell membranes, coenzyme Q, and other structures from free radical oxidation damage, thereby curbing the generation of toxic peroxidation products. It may also have a specific structural role in biological membranes.

Indications

Supplemental doses for patients at risk of vitamin E deficiency (e.g., neuromuscular diseases, neurological defects in hepatobiliary disease, haemolytic anaemia)G-6-PD deficiency (to increase survival time of erythrocytes)Acanthocytosis (to normalize oxidative fragility of erythrocytes)Reduction of retrolental fibroplasia risk in premature infantsAdjunct with vitamin A to enhance its absorption and storage, and to reduce toxicity in hypervitaminosis ASymptomatic improvement in intermittent claudication, fibrocystic breast disease, and nocturnal muscle cramps

Dosing

Adult
Supplemental doses: 10–30 mg/day. G-6-PD deficiency: 100 mg/day. Acanthocytosis: 100 mg/week i.m. Intermittent claudication, fibrocystic breast disease, nocturnal muscle cramps: 400–600 mg/day.
Pediatric
Retrolental fibroplasia in premature infants: 100 mg/kg/day oral.

Pharmacokinetics

Protein binding
Circulates in plasma in association with β-lipoprotein.
Metabolism
Circulates in plasma in association with β-lipoprotein, is stored in tissues.

Side effects

Common
Abdominal crampsLoose motionsLethargy
Serious
  • Creatinuria
  • Impaired wound healing

Drug interactions

Iron
Moderate
Textbook

Reduced effectiveness of iron therapy.

Monitor patients receiving concomitant vitamin E and iron therapy for the effectiveness of iron supplementation; adjustment of dosing schedules or amounts may be necessary.

Source: KDT 7e · p912

Related guidelines

Other Fat-soluble vitamin drugs

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Sources: KD Tripathi 7e·Verified: 2026-05-10 · House clinical team