Drug reference directory
Drug reference

urapidil

α1 receptor antagonist · Antihypertensive, Alpha Blocker

α1 receptor antagonistAntihypertensive, Alpha BlockerATC C02CA06
CDSCO approvedATC C02CA06
EXCRETION
—
not curated
INTERACTIONS
—
none in our sources
PREGNANCY
—
not curated

Mechanism

Urapidil is a selective α1 receptor antagonist that causes hypotension primarily through peripheral α1 adrenergic receptor blockade, but also has CNS actions.

Related guidelines

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Textbook-sourced·Sources: Goodman & Gilman 14e·Updated: 2026-05-10