Drug lookup
Drug reference

hexamethonium

Ganglionic blocking agent (Nn receptor antagonist) · Research tool (historical antihypertensive)

Ganglionic blocking agent (Nn receptor antagonist)Research tool (historical antihypertensive)
CDSCO approved
EXCRETION
not curated
INTERACTIONS
none in our sources
PREGNANCY
not curated

Mechanism

Blocks the channel after it opens, shortening the duration of current flow by either occluding the open channel or causing it to close. This blocks the initial EPSP and inhibits ganglionic transmission.

Side effects

Serious
  • Numerous undesirable side effects due to generalized ganglionic blockade

Related guidelines

Other Ganglionic blocking agent (Nn receptor antagonist) drugs

Ask House about hexamethonium

Continue into a citation-backed clinical answer with the drug context already attached.

Sources: Goodman & Gilman 14e·Verified: 2026-05-10 · House clinical team