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procaterol

β2-selective receptor agonist · Bronchodilator

β2-selective receptor agonistBronchodilatorATC R03AC08
CDSCO approvedATC R03AC08
EXCRETION
not curated
INTERACTIONS
7 major
SEVERE in our sources
PREGNANCY
not curated
Top interactionssee all 9
  • IsocarboxazidSevereTextbookG&G 14e · p264
  • MoclobemideSevereTextbookG&G 14e · p264
  • PhenelzineSevereTextbookG&G 14e · p264
  • ProcarbazineSevereTextbookG&G 14e · p264

Mechanism

Procaterol is a β2-selective receptor agonist with a prompt onset of action.

Pharmacokinetics

Onset
prompt onset of action (inhalation)
Protein binding
sustained for about 5 h (inhalation)

Drug interactions

Isocarboxazid
Severe
Textbook

Increased risk of adverse cardiovascular effects.

At least 2 weeks should elapse between the use of MAO inhibitors and administration of β2 agonists or other sympathomimetics.

Source: G&G 14e · p264

Moclobemide
Severe
Textbook

Increased risk of adverse cardiovascular effects.

At least 2 weeks should elapse between the use of MAO inhibitors and administration of β2 agonists or other sympathomimetics.

Source: G&G 14e · p264

Phenelzine
Severe
Textbook

Increased risk of adverse cardiovascular effects.

At least 2 weeks should elapse between the use of MAO inhibitors and administration of β2 agonists or other sympathomimetics.

Source: G&G 14e · p264

Procarbazine
Severe
Textbook

Increased risk of adverse cardiovascular effects.

At least 2 weeks should elapse between the use of MAO inhibitors and administration of β2 agonists or other sympathomimetics.

Source: G&G 14e · p264

Rasagiline
Severe
Textbook

Increased risk of adverse cardiovascular effects.

At least 2 weeks should elapse between the use of MAO inhibitors and administration of β2 agonists or other sympathomimetics.

Source: G&G 14e · p264

Selegiline
Severe
Textbook

Increased risk of adverse cardiovascular effects.

At least 2 weeks should elapse between the use of MAO inhibitors and administration of β2 agonists or other sympathomimetics.

Source: G&G 14e · p264

Tranylcypromine
Severe
Textbook

Increased risk of adverse cardiovascular effects.

At least 2 weeks should elapse between the use of MAO inhibitors and administration of β2 agonists or other sympathomimetics.

Source: G&G 14e · p264

Corticosteroids
Moderate
Textbook

Enhanced beneficial effects in asthma therapy for both drugs.

Source: G&G 14e · p887

Digoxin
Moderate
Textbook

Hypokalemia, which could predispose to cardiac arrhythmias, especially in patients with cardiac disease.

Use with caution.

Source: G&G 14e · p264

Related guidelines

Other β2-selective receptor agonist drugs

Ask House about procaterol

Continue into a citation-backed clinical answer with the drug context already attached.

Sources: Goodman & Gilman 14e·Verified: 2026-05-10 · House clinical team