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relacorilant

Selective glucocorticoid receptor antagonist · Glucocorticoid receptor antagonist

Selective glucocorticoid receptor antagonistGlucocorticoid receptor antagonist
CDSCO approved
EXCRETION
not curated
INTERACTIONS
none in our sources
PREGNANCY
not curated

Mechanism

An orally available, high-affinity, selective antagonist for the glucocorticoid receptor. Unlike mifepristone, it does not have appreciable affinity at the progesterone receptor.

Indications

endogenous cushing syndrome (under clinical trials)adrenocortical carcinoma (under clinical trials)

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Sources: Goodman & Gilman 14e·Verified: 2026-05-10 · House clinical team