Drug reference directory
Drug reference

relacorilant

Selective glucocorticoid receptor antagonist · Glucocorticoid receptor antagonist

Selective glucocorticoid receptor antagonistGlucocorticoid receptor antagonist
CDSCO approved
EXCRETION
—
not curated
INTERACTIONS
—
none in our sources
PREGNANCY
—
not curated

Mechanism

An orally available, high-affinity, selective antagonist for the glucocorticoid receptor. Unlike mifepristone, it does not have appreciable affinity at the progesterone receptor.

Indications

endogenous cushing syndrome (under clinical trials)adrenocortical carcinoma (under clinical trials)

Related guidelines

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Textbook-sourced·Sources: Goodman & Gilman 14e·Updated: 2026-05-10