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nitrendipine

Dihydropyridine calcium channel blocker · Antianginal

Dihydropyridine calcium channel blockerAntianginal
CDSCO approved
EXCRETION
not curated
INTERACTIONS
none in our sources
PREGNANCY
not curated

Mechanism

Releases NO from the endothelium and inhibits cAMP phosphodiesterase, contributing to vasodilator action. The endothelial NO may retard atherosclerosis. Does not depress ventricular contractility and A-V conduction.

Indications

HypertensionAngina pectoris

Dosing

Adult
5–20 mg OD

Pharmacokinetics

Half-life
4–12 hours
Bioavailability
10–30%

Drug interactions

Ursodeoxycholic Acid
Mild
Database

Potentially increased nitrendipine levels and risk of adverse effects (e.g., hypotension).

Monitor blood pressure and for nitrendipine-related adverse effects. Dose adjustment of nitrendipine may be needed.

Related guidelines

Other Dihydropyridine calcium channel blocker drugs

Ask House about nitrendipine

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Sources: KD Tripathi 7e·Verified: 2026-05-10 · House clinical team